RBFE network

Selected edges are shown below with both ligands drawn side by side. The warm highlight is the soft-core region that changes during the transformation; the cool highlight is the common core that stays fixed.

16
Ligands
44
Edges
11
Repaired
0
Rejected
optimal
Planner
Unmet constraints

Diagnostics

Network-level metrics. Machine time is estimated from published per-edge measurements and is a report only -- it played no part in choosing these edges.

MetricValue
Total cost221.039 scorer units
Estimated machine time174.7 GPU-hours (about $69.87)
Mean cost per edge5.024
Degreemin 1 · mean 5.50 · max 13
Isolated ligandsnone
Diameter3
Short cycles205 of length ≤ 4
Robustness91% of 100 trials stay connected at 5% edge failure; 15.9 ligands retained on average

44 edges over 16 ligands is 1 below the n*ln(n) precision floor of 45 (Pitman 2023). Below that floor precision degrades faster as the series grows; raise --edges-per-ligand or --n-edges to buy it back.

Network

ejm31 - ejm42: cost 4.345ejm31 - ejm44: cost 5.449ejm31 - ejm45: cost 5.182ejm31 - ejm46: cost 5.130ejm31 - ejm47: cost 5.449ejm31 - ejm48: cost 5.736ejm31 - ejm49: cost 5.999ejm31 - ejm50: cost 4.345ejm31 - ejm54: cost 5.130ejm31 - ejm55: cost 4.759ejm31 - jmc23: cost 5.449ejm31 - jmc27: cost 5.449ejm31 - jmc28: cost 5.449ejm42 - ejm43: cost 4.398ejm42 - ejm44: cost 5.449ejm42 - ejm45: cost 5.182ejm42 - ejm47: cost 5.449ejm42 - ejm50: cost 4.345ejm42 - ejm55: cost 4.759ejm42 - jmc23: cost 5.449ejm42 - jmc27: cost 5.449ejm42 - jmc28: cost 5.449ejm43 - ejm44: cost 4.449ejm43 - ejm45: cost 5.449ejm43 - ejm46: cost 5.130ejm43 - ejm54: cost 5.130ejm43 - ejm55: cost 5.130ejm45 - ejm50: cost 5.182ejm46 - ejm50: cost 5.130ejm46 - ejm54: cost 5.130ejm46 - ejm55: cost 5.130ejm46 - jmc23: cost 4.449ejm46 - jmc27: cost 4.449ejm46 - jmc28: cost 4.449ejm46 - jmc30: cost 4.914ejm50 - ejm54: cost 5.130ejm50 - ejm55: cost 4.759ejm54 - ejm55: cost 5.130jmc23 - jmc27: cost 4.449jmc23 - jmc28: cost 4.449jmc23 - jmc30: cost 4.914jmc27 - jmc28: cost 4.449jmc27 - jmc30: cost 4.914jmc28 - jmc30: cost 4.914ejm31 (degree 13)ejm31ejm31ejm42 (degree 10)ejm42ejm42ejm43 (degree 6)ejm43ejm43ejm44 (degree 3)ejm44ejm44ejm45 (degree 4)ejm45ejm45ejm46 (degree 9)ejm46ejm46ejm47 (degree 2)ejm47ejm47ejm48 (degree 1)ejm48ejm48ejm49 (degree 1)ejm49ejm49ejm50 (degree 6)ejm50ejm50ejm54 (degree 5)ejm54ejm54ejm55 (degree 6)ejm55ejm55jmc23 (degree 6)jmc23jmc23jmc27 (degree 6)jmc27jmc27jmc28 (degree 6)jmc28jmc28jmc30 (degree 4)jmc30jmc30

Thicker edges are cheaper. Hollow red nodes are unconnected. Click a network edge or the index below to jump to its transformation card.

Selected edges

soft-core (transformed)common core (held fixed)
ejm31~ejm42cost 4.345 · soft-core 1/4 · common core 31ejm31~ejm50cost 4.345 · soft-core 1/2 · common core 31ejm50~ejm42cost 4.345 · soft-core 2/4 · common core 31ejm42~ejm43cost 4.398 · soft-core 1/4 · common core 34ejm43~ejm44cost 4.449 · soft-core 1/4 · common core 37ejm46~jmc23cost 4.449 · soft-core 1/1 · common core 35ejm46~jmc27cost 4.449 · soft-core 1/1 · common core 35ejm46~jmc28cost 4.449 · soft-core 1/4 · common core 35jmc23~jmc27cost 4.449 · soft-core 1/1 · common core 35jmc23~jmc28cost 4.449 · soft-core 1/4 · common core 35jmc27~jmc28cost 4.449 · soft-core 1/4 · common core 35ejm31~ejm55cost 4.759 · soft-core 4/5 · common core 28ejm55~ejm42cost 4.759 · soft-core 5/7 · common core 28ejm50~ejm55cost 4.759 · soft-core 5/5 · common core 28ejm46~jmc30cost 4.914 · soft-core 1/2 · common core 35jmc23~jmc30cost 4.914 · soft-core 1/2 · common core 35jmc27~jmc30cost 4.914 · soft-core 1/2 · common core 35jmc30~jmc28cost 4.914 · soft-core 2/4 · common core 35ejm31~ejm46cost 5.130 · soft-core 4/8 · common core 28ejm31~ejm54cost 5.130 · soft-core 4/9 · common core 28ejm46~ejm43cost 5.130 · soft-core 8/10 · common core 28ejm54~ejm43cost 5.130 · soft-core 9/10 · common core 28ejm55~ejm43cost 5.130 · soft-core 5/10 · common core 28ejm50~ejm46cost 5.130 · soft-core 5/8 · common core 28ejm46~ejm54cost 5.130 · soft-core 8/9 · common core 28ejm55~ejm46cost 5.130 · soft-core 5/8 · common core 28ejm50~ejm54cost 5.130 · soft-core 5/9 · common core 28ejm55~ejm54cost 5.130 · soft-core 5/9 · common core 28ejm31~ejm45cost 5.182 · soft-core 1/8 · common core 31ejm42~ejm45cost 5.182 · soft-core 4/8 · common core 31ejm50~ejm45cost 5.182 · soft-core 2/8 · common core 31ejm31~ejm44cost 5.449 · soft-core 4/13 · common core 28ejm31~ejm47cost 5.449 · soft-core 4/11 · common core 28ejm31~jmc23cost 5.449 · soft-core 4/8 · common core 28ejm31~jmc27cost 5.449 · soft-core 4/8 · common core 28ejm31~jmc28cost 5.449 · soft-core 4/11 · common core 28ejm42~ejm44cost 5.449 · soft-core 7/13 · common core 28ejm42~ejm47cost 5.449 · soft-core 7/11 · common core 28ejm42~jmc23cost 5.449 · soft-core 7/8 · common core 28ejm42~jmc27cost 5.449 · soft-core 7/8 · common core 28ejm42~jmc28cost 5.449 · soft-core 7/11 · common core 28ejm43~ejm45cost 5.449 · soft-core 10/11 · common core 28ejm31~ejm48cost 5.736 · soft-core 4/14 · common core 28ejm31~ejm49cost 5.999 · soft-core 4/11 · common core 28

11 of the 11 repaired edges below can be toggled between the repaired soft-core and the one the mapper proposed. The repaired view is what is shown.

ejm31~ejm42

cost 4.345 · soft-core 1/4 · common core 31 · mapper mcss-e2

ejm31~ejm50

cost 4.345 · soft-core 1/2 · common core 31 · mapper mcss-e2

ejm50~ejm42

cost 4.345 · soft-core 2/4 · common core 31 · mapper mcss-e2
Soft-core repaired: regions (1, 1) → (1, 1), 2 atom(s) demoted.
(orientation flipped: sides below refer to ejm42~ejm50) closure: normalised raw soft-core 3/1 -> 4/2 atoms initial: 1 soft-core region(s) on side 1, 1 on side 2 final: 1/1 region(s), soft-core 4/2 atom(s)

ejm42~ejm43

cost 4.398 · soft-core 1/4 · common core 34 · mapper mcss-e2

ejm43~ejm44

cost 4.449 · soft-core 1/4 · common core 37 · mapper mcss-e2

ejm46~jmc23

cost 4.449 · soft-core 1/1 · common core 35 · mapper mcss-e2

ejm46~jmc27

cost 4.449 · soft-core 1/1 · common core 35 · mapper mcss-e2

ejm46~jmc28

cost 4.449 · soft-core 1/4 · common core 35 · mapper mcss-e2

jmc23~jmc27

cost 4.449 · soft-core 1/1 · common core 35 · mapper mcss-e2

jmc23~jmc28

cost 4.449 · soft-core 1/4 · common core 35 · mapper mcss-e2

jmc27~jmc28

cost 4.449 · soft-core 1/4 · common core 35 · mapper mcss-e2

ejm31~ejm55

cost 4.759 · soft-core 4/5 · common core 28 · mapper mcss-e2

ejm55~ejm42

cost 4.759 · soft-core 5/7 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (1, 1) → (1, 1), 8 atom(s) demoted.
(orientation flipped: sides below refer to ejm42~ejm55) initial: 1 soft-core region(s) on side 1, 1 on side 2 iter 1 side 1: absorbed 4 core atom(s) [31, 32, 33, 34] stranded behind the soft-core iter 1 side 2: absorbed 4 core atom(s) [29, 30, 31, 32] stranded behind the soft-core final: 1/1 region(s), soft-core 7/5 atom(s)

ejm50~ejm55

cost 4.759 · soft-core 5/5 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (1, 1) → (1, 1), 2 atom(s) demoted.
closure: normalised raw soft-core 4/4 -> 5/5 atoms initial: 1 soft-core region(s) on side 1, 1 on side 2 final: 1/1 region(s), soft-core 5/5 atom(s)

ejm46~jmc30

cost 4.914 · soft-core 1/2 · common core 35 · mapper mcss-e2

jmc23~jmc30

cost 4.914 · soft-core 1/2 · common core 35 · mapper mcss-e2

jmc27~jmc30

cost 4.914 · soft-core 1/2 · common core 35 · mapper mcss-e2

jmc30~jmc28

cost 4.914 · soft-core 2/4 · common core 35 · mapper mcss-e2

ejm31~ejm46

cost 5.130 · soft-core 4/8 · common core 28 · mapper mcss-e2

ejm31~ejm54

cost 5.130 · soft-core 4/9 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (1, 1) → (1, 1), 2 atom(s) demoted.
closure: normalised raw soft-core 3/8 -> 4/9 atoms initial: 1 soft-core region(s) on side 1, 1 on side 2 final: 1/1 region(s), soft-core 4/9 atom(s)

ejm46~ejm43

cost 5.130 · soft-core 8/10 · common core 28 · mapper mcss-e2

ejm54~ejm43

cost 5.130 · soft-core 9/10 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (2, 2) → (1, 1), 8 atom(s) demoted.
(orientation flipped: sides below refer to ejm43~ejm54) closure: normalised raw soft-core 6/5 -> 7/6 atoms initial: 2 soft-core region(s) on side 1, 2 on side 2 iter 1 side 1: bridged 2 regions by demoting 1 atom(s) [34] iter 1 side 2: bridged 2 regions by demoting 1 atom(s) [30] iter 1 side 1: absorbed 2 core atom(s) [35, 37] stranded behind the soft-core iter 1 side 2: absorbed 2 core atom(s) [31, 32] stranded behind the soft-core final: 1/1 region(s), soft-core 10/9 atom(s)

ejm55~ejm43

cost 5.130 · soft-core 5/10 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (1, 1) → (1, 1), 8 atom(s) demoted.
(orientation flipped: sides below refer to ejm43~ejm55) initial: 1 soft-core region(s) on side 1, 1 on side 2 iter 1 side 1: absorbed 4 core atom(s) [34, 35, 36, 37] stranded behind the soft-core iter 1 side 2: absorbed 4 core atom(s) [29, 30, 31, 32] stranded behind the soft-core final: 1/1 region(s), soft-core 10/5 atom(s)

ejm50~ejm46

cost 5.130 · soft-core 5/8 · common core 28 · mapper mcss-e2

ejm46~ejm54

cost 5.130 · soft-core 8/9 · common core 28 · mapper mcss-e2

ejm55~ejm46

cost 5.130 · soft-core 5/8 · common core 28 · mapper mcss-e2

ejm50~ejm54

cost 5.130 · soft-core 5/9 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (1, 1) → (1, 1), 4 atom(s) demoted.
closure: normalised raw soft-core 3/7 -> 5/9 atoms initial: 1 soft-core region(s) on side 1, 1 on side 2 final: 1/1 region(s), soft-core 5/9 atom(s)

ejm55~ejm54

cost 5.130 · soft-core 5/9 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (2, 2) → (1, 1), 6 atom(s) demoted.
(orientation flipped: sides below refer to ejm54~ejm55) initial: 2 soft-core region(s) on side 1, 2 on side 2 iter 1 side 1: bridged 2 regions by demoting 1 atom(s) [30] iter 1 side 2: bridged 2 regions by demoting 1 atom(s) [29] iter 1 side 1: absorbed 2 core atom(s) [31, 32] stranded behind the soft-core iter 1 side 2: absorbed 2 core atom(s) [30, 31] stranded behind the soft-core final: 1/1 region(s), soft-core 9/5 atom(s)

ejm31~ejm45

cost 5.182 · soft-core 1/8 · common core 31 · mapper mcss-e2

ejm42~ejm45

cost 5.182 · soft-core 4/8 · common core 31 · mapper mcss-e2

ejm50~ejm45

cost 5.182 · soft-core 2/8 · common core 31 · mapper mcss-e2

ejm31~ejm44

cost 5.449 · soft-core 4/13 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (3, 3) → (1, 1), 2 atom(s) demoted.
initial: 3 soft-core region(s) on side 1, 3 on side 2 iter 1 side 1: bridged 3 regions by demoting 1 atom(s) [19] [steiner:approximate] iter 1 side 2: bridged 3 regions by demoting 1 atom(s) [19] [steiner:approximate] final: 1/1 region(s), soft-core 4/13 atom(s)

ejm31~ejm47

cost 5.449 · soft-core 4/11 · common core 28 · mapper mcss-e2

ejm31~jmc23

cost 5.449 · soft-core 4/8 · common core 28 · mapper mcss-e2

ejm31~jmc27

cost 5.449 · soft-core 4/8 · common core 28 · mapper mcss-e2

ejm31~jmc28

cost 5.449 · soft-core 4/11 · common core 28 · mapper mcss-e2

ejm42~ejm44

cost 5.449 · soft-core 7/13 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (2, 2) → (1, 1), 10 atom(s) demoted.
initial: 2 soft-core region(s) on side 1, 2 on side 2 iter 1 side 1: bridged 2 regions by demoting 1 atom(s) [19] iter 1 side 2: bridged 2 regions by demoting 1 atom(s) [19] iter 1 side 1: absorbed 4 core atom(s) [31, 32, 33, 34] stranded behind the soft-core iter 1 side 2: absorbed 4 core atom(s) [37, 38, 39, 40] stranded behind the soft-core final: 1/1 region(s), soft-core 7/13 atom(s)

ejm42~ejm47

cost 5.449 · soft-core 7/11 · common core 28 · mapper mcss-e2

ejm42~jmc23

cost 5.449 · soft-core 7/8 · common core 28 · mapper mcss-e2

ejm42~jmc27

cost 5.449 · soft-core 7/8 · common core 28 · mapper mcss-e2

ejm42~jmc28

cost 5.449 · soft-core 7/11 · common core 28 · mapper mcss-e2

ejm43~ejm45

cost 5.449 · soft-core 10/11 · common core 28 · mapper mcss-e2
Soft-core repaired: regions (2, 2) → (1, 1), 4 atom(s) demoted.
initial: 2 soft-core region(s) on side 1, 2 on side 2 iter 1 side 1: bridged 2 regions by demoting 1 atom(s) [19] iter 1 side 2: bridged 2 regions by demoting 1 atom(s) [19] iter 1 side 1: absorbed 1 core atom(s) [29] stranded behind the soft-core iter 1 side 2: absorbed 1 core atom(s) [29] stranded behind the soft-core final: 1/1 region(s), soft-core 10/11 atom(s)

ejm31~ejm48

cost 5.736 · soft-core 4/14 · common core 28 · mapper mcss-e2

ejm31~ejm49

cost 5.999 · soft-core 4/11 · common core 28 · mapper mcss-e2